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LA REGINA
Si avvisano tutti gli studenti interessati che le lezioni del corso di Analisi Chimico Farmaceutica e Tossicologica I (M-Z) per l’anno accademico 2021/2022 avranno inizio lunedì 4 ottobre 2021 e proseguiranno con il seguente orario:
- lunedì 16:00 - 18:00, Aula Vincenzo Carelli, edificio CU019, link Google Meet: https://meet.google.com/zjn-otux-obz;
- martedì 11:00 - 13:00, Aula A, edificio CU018, link Google Meet: https://meet.google.com/stf-rhyu-gvt;
- mercoledì 16:00 - 18:00, Aula A - Raffaele Giuliano, edificio CU019, link Google Meet: https://meet.google.com/gpk-gvfw-sqo.
Ulteriori informazioni relative al corso possono essere reperite sul sito web dello stesso al link: https://elearning.uniroma1.it/course/view.php?id=461.
Previo appuntamento da concordare via email
| Course | Code | Year | Course - Attendance |
|---|---|---|---|
| PHARMACEUTICAL AND TOXICOLOGICAL ANALYTICAL CHEMISTRY I | 1022761 | 2021/2022 | Pharmaceutical Chemistry and Technology |
| PHARMACEUTICAL AND TOXICOLOGICAL ANALYTICAL CHEMISTRY I | 1022761 | 2020/2021 | Pharmaceutical Chemistry and Technology |
| PHARMACEUTICAL AND TOXICOLOGICAL ANALYTICAL CHEMISTRY I | 1022761 | 2019/2020 | Pharmaceutical Chemistry and Technology |
| PHARMACEUTICAL AND TOXICOLOGICAL ANALYTICAL CHEMISTRY I | 1022761 | 2018/2019 | Pharmaceutical Chemistry and Technology |
| PHARMACEUTICAL AND TOXICOLOGICAL ANALYTICAL CHEMISTRY I | 1022761 | 2017/2018 | Pharmaceutical Chemistry and Technology |
| PHARMACEUTICAL AND TOXICOLOGICAL ANALYTICAL CHEMISTRY I | 1022761 | 2016/2017 | Pharmaceutical Chemistry and Technology |
| Title | Journal | Year |
|---|---|---|
| Discovery of pyrrole derivatives for the treatment of glioblastoma and chronic myeloid leukemia | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | 2021 |
| Selenotriapine - an isostere of the most studied thiosemicarbazone with pronounced pro-apoptotic activity, low toxicity and ability to challenge phenotype reprogramming of 3-D mammary adenocarcinoma tumors | ARABIAN JOURNAL OF CHEMISTRY | 2020 |
| Discovery of new 1,1'-biphenyl-4-sulfonamides as selective subnanomolar human carbonic anhydrase II inhibitors | ACS MEDICINAL CHEMISTRY LETTERS | 2020 |
| Structure-activity relationship studies and in vitro and in vivo anticancer activity of novel 3-aroyl-1,4-diarylpyrroles against solid tumors and hematological malignancies | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | 2020 |
| Discovery of Zika virus NS2B/NS3 inhibitors that prevent mice from fife-threatening infection and brain damage | ACS MEDICINAL CHEMISTRY LETTERS | 2020 |
| New indolylarylsulfone non-nucleoside reverse transcriptase inhibitors show low nanomolar inhibition of single and double HIV-1 mutant strains | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | 2020 |
| Sulfonamide inhibitors of beta-Catenin signaling as anticancerAgents with different output on c-Myc | CHEMMEDCHEM | 2020 |
| Targeting the interaction between the SH3 domain of Grb2 and Gab2 | CELLS | 2020 |
| A new case manager for diabetic patients: a pilot observational study of the role of community pharmacists and pharmacy services in the case management of diabetic patients | PHARMACY | 2020 |
| Drug design and synthesis of first in class PDZ1 targeting NHERF1 inhibitors as anticancer agents | ACS MEDICINAL CHEMISTRY LETTERS | 2019 |
| Towards modern anticancer agents that interact with tubulin | EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES | 2019 |
| Small molecule inhibitors of KDM5 histone demethylases increase the radiosensitivity of breast cancer cells overexpressing Jarid1b | MOLECULES | 2019 |
| Switching on the activity of 1,5-diaryl-pyrrole derivatives against drug-resistant ESKAPE bacteria: structure-activity relationships and mode of action studies | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | 2019 |
| Bax activation blocks self-renewal and induces apoptosis of human glioblastoma stem cells | ACS CHEMICAL NEUROSCIENCE | 2018 |
| A negative allosteric modulator of WNT receptor frizzled 4 switches into an allosteric agonist | BIOCHEMISTRY | 2018 |
| β-catenin knockdown promotes nherf1-mediated survival of colorectal cancer cells: implications for a double-targeted therapy | ONCOGENE | 2018 |
| New 6- and 7-heterocyclyl-1H-indole derivatives as potent tubulin assembly and cancer cell growth inhibitors | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | 2018 |
| Treating chronic myeloid leukemia by inhibition of tubulin polymerization | 2018 | |
| Structure-based drug design of potent pyrazole derivatives against Rhinovirus replication | JOURNAL OF MEDICINAL CHEMISTRY | 2018 |
| DOACs: aspetti chimico-farmaceutici e tossicologici | 2018 |
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Teaching materials
Department
CHIMICA E TECNOLOGIE DEL FARMACO
SSD
CHIM/08